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CTP354
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CTP354图片
规格:98%
分子量:408.5
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议

产品介绍
A deuterated derivative of L-838,417
货号:ajcx28338
CAS:1213669-91-0
分子式:C19H10D9F2N7O
分子量:408.5
溶解度:DMF: 3 mg/ml,DMSO: 3 mg/ml,Ethanol: 2 mg/ml,PBS (pH 7.2): insol
纯度:98%
存储:Store at -20°C
库存:现货

Background:

CTP354 is a deuterated derivative of the GABAAreceptor modulator L-838,417.1It binds to the GABAAreceptor benzodiazepine binding site in non-α1subunit-containing GABAAreceptors. CTP354 has a longer duration of action than L-838,417 in a rat model of neuropathic pain induced by sciatic nerve ligation.

1.Harbeson, S.L., and Tung, R.D.Deuterium medicinal chemistry: A new approach to drug discovery and developmentMedchem News24(2)8-22(2014)