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L 689502
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CAS NO:138483-63-3
包装:50mg, 100mg, 250mg
规格:≥98%

产品介绍

L 689502 is a potent inhibitor of HIV-l protease with an IC50 of 1 nM. IC50 & 1 nM (HIV-l protease) Both L694746 and L-689502 inhibit HIV-l ptotease activity in a concentration-dependent manner. Pepstatin is much less potent than either compound exhibiting an IC50 of 2 μM. L694746 is as potent as L-689502 in inhibiting the HIV-l protease despite being structurally different from L-689502. References: Vieth M, Cummins DJ. DoMCoSAR: a novel approach for establishing the docking mode that is consistent with the structure-activity relationship. Application to HIV-1 protease inhibitors and VEGF receptor tyrosine kinase inhibitors. J Med Chem. 2000 Aug 10;43(16):3020-32. PubMed PMID: 10956210.

纯度:≥98%

CAS:138483-63-3