GSK-554418A is a novel azaindole CB(2) agonists. GSK-554418A is used for the treatment of chronic pain. This compound was efficacious in the acute model and the chronic joint pain model. References: Giblin GM, Billinton A, Briggs M, Brown AJ, Chessell IP, Clayton NM, Eatherton AJ, Goldsmith P, Haslam C, Johnson MR, Mitchell WL, Naylor A, Perboni A, Slingsby BP, Wilson AW. Discovery of 1-[4-(3-chlorophenylamino)-1-methyl-1H-pyrrolo[3,2-c]pyridin-7-yl]-1-morpholin-4- ylmethanone (GSK554418A), a brain penetrant 5-azaindole CB2 agonist for the treatment of chronic pain. J Med Chem. 2009 Oct 8;52(19):5785-8. doi: 10.1021/jm9009857. PubMed PMID: 19743867.

纯度：≥98%

CAS：871819-90-8