G-15, formerly known as GRB-G15, is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM). References: Imesch P, Samartzis EP, Dedes KJ, Fink D, Fedier A. Histone deacetylase inhibitors down-regulate G-protein-coupled estrogen receptor and the GPER-antagonist G-15 inhibits proliferation in endometriotic cells. Fertil Steril. 2013 Sep;100(3):770-6. doi: 10.1016/j.fertnstert.2013.05.008. Epub 2013 Jun 10. PubMed PMID: 23755949.
纯度:≥98%
CAS:1161002-05-6