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GlyH-101
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
GlyH-101图片
CAS NO:328541-79-3
规格:≥98%
包装与价格:
包装价格(元)
2mg电议
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议
250mg电议
500mg电议

产品介绍

GlyH-101 is a novel and potent CFTR inhibitor (cystic fibrosis transmembrane conductance regulator) with Ki of 1.4 uM. GlyH-101 is a glycine hydrazide that has been shown to block CFTR channels. GlyH-101 blocked I(Cl.PKA) in a concentration- and voltage-dependent fashion (IC(50) at +100 mV=0.3 A± 1.5 μM and at -100 mV=5.1 A± 1.3 μM). GlyH-101 blocks the open pore of cardiac CFTR channels at an electrical distance of 0.15 A± 0.03 from the external membrane surface.

纯度:≥98%

CAS:328541-79-3