GI-530159 is a selective dual trek1 and trek2 channel activator References: Loucif AJC, Saintot PP, Liu J, Antonio BM, Zellmer SG, Yoger K, Veale EL, Wilbrey A, Omoto K, Cao L, Gutteridge A, Castle NA, Stevens EB, Mathie A. GI-530159, a novel, selective, mechanosensitive two-pore-domain potassium (K(2P) ) channel opener, reduces rat dorsal root ganglion neuron excitability. Br J Pharmacol. 2018 Jun;175(12):2272-2283. doi: 10.1111/bph.14098. Epub 2017 Dec 29. PubMed PMID: 29150838; PubMed Central PMCID: PMC5980259.
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