DA-3934 is of phenoxyacetanilide analogues, it has high affinity for gastrin/CCK-B receptors and high selectivity over CCK-A receptors. DA-3934 and its methyl ester analogue inhibited pentagastrin-induced gastric acid secretion in rats in a dose-dependent manner. References: Takeda Y, Kawagoe K, Yokomizo A, Yokomizo Y, Hosokami T, Shimoto Y, Tabuchi Y, Ogihara Y, Otsubo R, Honda Y, Yokohama S. Synthesis of phenoxyacetic acid derivatives as highly potent antagonists of gastrin/cholecystokinin-B receptors. II. Chem Pharm Bull (Tokyo). 1998 Jun;46(6):951-61. PubMed PMID: 9658573.
纯度:≥98%
CAS:183176-50-3