Dexisometheptene is an antimigraine drug candidate. The active ingredient in TNX-201 is dexisometheptene mucate, the (R) isomer of isometheptene mucate. TNX-201 significantly increases the pain threshold of acute pain response, and potently and selectively binds to receptors in the central nervous system known as imidazoline type-1 (I1) receptors, where it acts as a receptor agonist. References:

纯度：≥98%

CAS：1620401-56-0