CGP 20712A Dihydrochoride is a potent and selective antagonist of β1-adrenoceptor with IC50 of 0.7 nM . References: Janssens K, Boussemaere M, Wagner S, Kopka K, Denef C. Beta1-adrenoceptors in rat anterior pituitary may be constitutively active. Inverse agonism of CGP 20712A on basal 3',5'-cyclic adenosine 5'-monophosphate levels. Endocrinology. 2008 May;149(5):2391-402. doi: 10.1210/en.2007-1397. PubMed PMID: 18202135.
纯度:≥98%
CAS:1216905-73-5