CGP-54626 is a selective antagonist of the GABAB receptor with an IC50 of 4 nM.1 It can be used to investigate the role of GABAB receptors in neurological signaling. References: Wood MD, Murkitt KL, Rice SQ, Testa T, Punia PK, Stammers M, Jenkins O, Elshourbagy NA, Shabon U, Taylor SJ, Gager TL, Minton J, Hirst WD, Price GW, Pangalos M. The human GABA(B1b) and GABA(B2) heterodimeric recombinant receptor shows low sensitivity to phaclofen and saclofen. Br J Pharmacol. 2000 Nov;131(6):1050-4. PubMed PMID: 11082110; PubMed Central PMCID: PMC1572438.

纯度：≥98%

CAS：149936-58-3