CP-199330 is a cysteinyl LT1 receptor antagonist that is equipotent to marketed cysLT1 receptor antagonists zafirlukast and pranlukas. It is devoid of liver toxicity. References: Chambers RJ, Marfat A, Antognoli GW, Cheng JB, Damon DB, Kuperman AV, Liston TC, Mebus C, Pillar JS, Shirley JT, Watson JW. Discovery of CP-199,330 and CP-199,33 two potent and orally efficacious cysteinyl LT1 receptor antagonists devoid of liver toxicity. Bioorg Med Chem Lett. 1999 Sep 20;9(18):2773-8. PubMed PMID: 10509933.
纯度:≥98%
CAS:158102-92-2