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Itacnosertib
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Itacnosertib图片
CAS NO:1628870-27-8
包装与价格:
包装价格(元)
10mM*1 mL电议
5mg电议
10mg电议
25mg电议
50mg电议

产品介绍
Itacnosertib (TP-0184) 是JAK2,ACVR1 (ALK2)和ALK5的抑制剂,如WO2014151871所述。
Cas No.1628870-27-8
别名TP-0184
分子式C26H28N8O
分子量468.55
溶解度DMSO : 12.5 mg/mL (26.68 mM; ultrasonic and warming and heat to 60°C)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Itacnosertib (TP-0184) is both inhibitor to JAK2, ACVR1 (ALK2) and ALK5 as described in WO2014151871[1].

[1]. Mollard, Alexis; Warner, Steven L.; Flynn, Gary A.; Vankayalapati, Hariprasad; Bearss, David J. Preparation of [(piperazinylphenyl)amino]pyrimidine derivatives as JAK2 and ALK2 inhibitors. WO2014151871 A2