EP3 antagonist 3 (compound 2) 是一种口服有效的、选择性的 EP3 拮抗剂,其 pKi 为 8.3。EP3 antagonist 3 具有良好的药代动力学特性。EP3 antagonist 3 可用于膀胱过度活动症 (OAB) 的研究。
Cas No. | 1227827-88-4 |
分子式 | C21H18N2O4 |
分子量 | 362.38 |
溶解度 | DMSO : 250 mg/mL (689.88 mM; Need ultrasonic) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | EP3 antagonist 3 (compound 2) is an orally active, potent and selectiveEP3antagonist, with apKiof 8.3. EP3 antagonist 3 shows excellent pharmacokinetic properties. EP3 antagonist 3 can be used for overactive bladder (OAB) research[1]. |