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CAY10788
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CAY10788图片
CAS NO:119515-00-3
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议
25mg电议

产品介绍
A CysLT1receptor antagonist
Cas No.119515-00-3
Canonical SMILESO=C(OC)C1=CC(OCC2=NC3=CC=CC=C3C=C2)=CC=C1
分子式C18H15NO3
分子量293.3
溶解度DMF: insol,DMSO: 1 mg/ml,Ethanol: 1 mg/ml,PBS (pH 7.2): insol
储存条件-20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

CAY10788 is an antagonist of the cysteinyl leukotriene 1 (CysLT1) receptor (IC50= 3.9 µM).1

1.Fiorillo, B., Sepe, V., Conflitti, P., et al.Structural basis for developing multitarget compounds acting on cysteinyl leukotriene receptor 1 and G-protein-coupled bile acid receptor 1J. Med. Chem.64(22)16512-16529(2021)