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AGN 205327
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
AGN 205327图片
包装与价格:
包装价格(元)
2mg电议
5mg电议
10mg电议

产品介绍
AGN 205327是RAR激动剂,对RARα/β/γ的EC50分别为3766/734/32 nM,对RXR无抑制性。
Canonical SMILESCC1(C)CCC(C)(C)C2=C1C=CC(/C(C3=CC4=CC(C(O)=O)=CC=C4N3)=N\O)=C2
分子式C24H26N2O3
分子量390.47
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

AGN 205327 is a potent synthetic RARs agonist with EC50 of 3766/734/32 nM for RARα/β/γ respectively; no inhibition on RXR.IC50 value: 3766/734/32 nM for RARα/β/γTarget: RAR agonist

[1]. Preferential binding of synthetic retinoid analogs to subtypes of RAR.