包装 | 价格(元) |
1mg | 电议 |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
Canonical SMILES | O=C(CNC(C[C@@H](C(O)=O)NC([C@@H](C1=CC=CC=C1)NC([C@H]2CCCCN)=O)=O)=O)N[C@@H](CCCNC(N)=N)C(N2C)=O.OC(C(F)(F)F)=O |
分子式 | C29H42F3N9O9 |
分子量 | 717.69 |
溶解度 | DMSO: 250 mg/mL (348.34 mM) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | c(phg-isoD-G-R-(NMe)k) TFA is a selective and potent α5β1-integrin ligand with an IC50 of 2.9 nM[1]. c(phg-isoD-G-R-(NMe)k) TFA is trimerized with the chelator TRAP and used as a positron-emission tomography tracer for monitoring α5β1 integrin expression in a M21 mouse xenograft[1]. [1]. Kapp TG, et al. N-Methylation of isoDGR Peptides: Discovery of a Selective α5β1-Integrin Ligand as a Potent Tumor Imaging Agent. J Med Chem. 2018 Mar 22;61(6):2490-2499. |