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Didesmethyl cariprazine
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Didesmethyl cariprazine图片
CAS NO:839712-25-3
包装:5mg
市场价:4950元

产品介绍
Didesmethyl cariprazine 是 Cariprazine 的代谢物，作为主要的循环活性部分。Didesmethyl cariprazine 的半衰期较长，为 1-3 周。Cariprazine是一种新型抗精神病候选药物，能结合 D3, D2 和 5-HT1A 。
Cas No.839712-25-3
分子式C19H28Cl2N4O
分子量399.36
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic drug candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor[1].

[1]. Citrome L, et al. Cariprazine for acute and maintenance treatment of adults with schizophrenia: an evidence-based review and place in therapy. Neuropsychiatr Dis Treat. 2018 Oct 5;14:2563-2577.