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Methyl-6-alpha-Naltrexol
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Methyl-6-alpha-Naltrexol图片
CAS NO:116388-85-3
包装:1mg
市场价:3600元

产品介绍
Methyl-6-alpha-Naltrexol 是甲基纳曲酮 (MNTX) 的代谢物 (metabolite)。Methyl-6-alpha-Naltrexol 是一种选择性的 mu-阿片受体 (mu-opioid receptor) 拮抗剂,在胃肠道组织中起外周作用的受体拮抗剂作用。
Cas No.116388-85-3
分子式C21H27NO4
分子量357.44
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Methyl-6-alpha-Naltrexol is a metabolite of Methylnaltrexone (MNTX). Methylnaltrexone is a selective mu-opioid receptor antagonist and functions as a peripherally acting receptor antagonist in tissues of the gastrointestinal tract[1].

[1]. Appavu Chandrasekaran,et al. Metabolism of intravenous methylnaltrexone in mice, rats, dogs, and humans. Drug Metab Dispos. 2010 Apr;38(4):606-16.