CAS NO: | 1276124-00-5 |
包装 | 价格(元) |
5mg | 电议 |
10mM (in 1mL Water) | 电议 |
25mg | 电议 |
50mg | 电议 |
100mg | 电议 |
Cas No. | 1276124-00-5 |
别名 | 内吗啡肽 2 三氟乙酸盐 |
Canonical SMILES | O=C(N)[C@H](CC1=CC=CC=C1)NC([C@H](CC2=CC=CC=C2)NC([C@H]3N(C([C@H](CC4=CC=C(C=C4)O)N)=O)CCC3)=O)=O.OC(C(F)(F)F)=O |
分子式 | C34H38F3N5O7 |
分子量 | 685.69 |
溶解度 | Water: 62.5 mg/mL (91.15 mM); DMSO:< 1 mg/mL (insoluble or slightly soluble) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1]. Ki: 20-30 nM (kappa3 opioid receptor)[1] [1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13. |