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Paliperidone palmitate
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Paliperidone palmitate图片
CAS NO:199739-10-1
包装:10mg
市场价:630元

产品介绍
Paliperidonepalmitate(9-Hydroxyrisperidonepalmitate)是一种非典型长效抗精神病药，是Paliperidone的酯类前药。Paliperidone是一种非典型抗精神病药的多巴胺(dopamine)拮抗剂和5-HT2A拮抗剂。Paliperidonepalmitate对精神分裂症有效。
Cas No.199739-10-1
别名棕榈酸帕利哌酮,9-Hydroxyrisperidone palmitate
Canonical SMILESO=C(OC1CCCN(C1=NC(C)=C2CCN3CCC(C4=NOC5=C4C=CC(F)=C5)CC3)C2=O)CCCCCCCCCCCCCCC
分子式C39H57FN4O4
分子量664.89
储存条件4℃, away from moisture and light
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Paliperidone palmitate (9-Hydroxyrisperidone palmitate), an atypical long-acting antipsychotic agent, is an ester prodrug of Paliperidone. Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class. Paliperidone palmitate shows efficacy against schizophrenia[1].

[1]. Kwon JS, et al. Satisfaction of immediate or delayed switch to paliperidone palmitate in patients unsatisfied with current oral atypical antipsychotics. Int Clin Psychopharmacol. 2015;30(6):320-328.