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TC-G 1003
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
TC-G 1003图片
CAS NO:1021912-42-4
包装:10mg
市场价:4013元

产品介绍
TC-G 1003 是一种有效的生长抑素受体亚型 2 (sst2) 激动剂,其 Ki 值为 0.025 nM,cAMP IC50 值为 4.8 nM。
Cas No.1021912-42-4
Canonical SMILESCC1=CC(C3=C(OCCCN)C2=CC(C4=CC=CC(O)=C4)=C(Cl)C=C2N=C3)=CC(C)=C1
分子式C26H25ClN2O2
分子量432.94
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

High affinity somatostatin sst2 receptor agonist (Ki = 0.025 nM). Inhibits growth hormone secretion and attenuates laser-induced ocular neovascular lesion size in rats.

Wolkenberg et al (2011) Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2. J.Med.Chem. 54 2351 PMID:21395312