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Glutaminase-IN-3
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Glutaminase-IN-3图片
CAS NO:1439399-45-7
包装与价格:
包装价格(元)
10mM (in 1mL DMSO)电议
50mg电议
100mg电议

产品介绍
Glutaminase-IN-3 (compound 657) 是一种有效的 glutaminase 抑制剂,对GLS1的 IC50 值为0.24 μM。详细情况请参见专利 WO2014089048A1,compound 657。
Cas No.1439399-45-7
别名N-[6-[4-(5-氨基-1,3,4-噻二唑-2-基)丁基]-3-哒嗪基]-3-(三氟甲氧基)苯乙酰胺
分子式C19H19F3N6O2S
分子量452.45
溶解度DMSO : 50 mg/mL (110.51 mM; Need ultrasonic)
储存条件4°C, protect from light
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Glutaminase-IN-3 (compound 657) is a potent glutaminase inhibitor with an IC50 of 0.24 μM for Glutaminase 1 (GLS1). Glutaminase-IN-3 is extracted from patent WO2014089048A1, compound 657[1].

[1]. Mark K. Bennett, et al. Treatment of cancer with heterocyclic inhibitors of glutaminase. WO2014089048A1.