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LPA2 antagonist 2
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
LPA2 antagonist 2图片
CAS NO:36840-10-5
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议
50mg电议
100mg电议

产品介绍
LPA2 antagonist 2 (H2L 5226501) 是一种选择性 LPA2 拮抗剂,IC50 为 28.3 nM,比 LPA3 (IC50 为 13.85 μM) 选择性高 480 倍以上。
Cas No.36840-10-5
Canonical SMILESO=C(O)/C=C/C(NC1=CC=C(C2=CC=C(NC(/C=C/C(O)=O)=O)C=C2)C=C1)=O
分子式C20H16N2O6
分子量380.35
溶解度DMSO: 83.33 mg/mL (219.09 mM)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is >480-fold more selective than LPA3 (IC50 of 13.85 μM)[1].

[1]. Fells JI, et al. Identification of non-lipid LPA3 antagonists by virtual screening. Bioorg Med Chem. 2008 Jun 1;16(11):6207-17.