CAS NO: | 1202235-68-4 |
包装 | 价格(元) |
10mM (in 1mL DMSO) | 电议 |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
200mg | 电议 |
500mg | 电议 |
Cas No. | 1202235-68-4 |
Canonical SMILES | O=C1NC(C(O)=CC=C2C(O)CNC(C)(CC3=C(C=CC=C3)C)C)=C2OC1 |
分子式 | C21H26N2O4 |
分子量 | 370.44 |
溶解度 | DMSO: 75 mg/mL (202.46 mM) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM[1]. Compared to other βAR ligands, BI-167107 displays nanomolar affinities and slow off-rates[1]. [1]. Rasmussen SG, et al. Structure of a nanobody-stabilized active state of the β(2) adrenoceptor. Nature. 2011 Jan 13;469(7329):175-80. |