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Bilaid A
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Bilaid A图片
CAS NO:2393865-97-7
包装与价格：
包装价格(元)
1mg电议
5mg电议

产品介绍
A tetrapeptide µ-opioid receptor agonist
Cas No.2393865-97-7
Canonical SMILESO=C(N[C@H](C(C)C)C(N[C@@H](C(C)C)C(N[C@H](CC1=CC=CC=C1)C(O)=O)=O)=O)[C@@H](N)CC2=CC=CC=C2
分子式C28H38N4O5
分子量510.6
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Bilaid A is a tetrapeptide agonist of the μ-opioid receptor (Ki= 3.1 μM using HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation in HEK293 cells expressing the human μ-opioid receptor by 21% when used at a concentration of 10 μM.

1.Dekan, Z., Sianati, S., Yousuf, A., et al.A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptorProc. Natl. Acad. Sci. USA116(44)22353-22358(2019)