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Cyproheptadine(hydrochloride hydrate)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Cyproheptadine(hydrochloride hydrate)图片
CAS NO:41354-29-4
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议
1g电议

产品介绍
Cyproheptadine (hydrochloride hydrate) 是一种抗组胺药,是血清素和组胺的拮抗剂2。
Cas No.41354-29-4
别名盐酸赛庚啶半水合物
Canonical SMILESCN(CC/1)CCC1=C2C(C=CC=C3)=C3C=CC4=C\2C=CC=C4.CN(CC/5)CCC5=C6C(C=CC=C7)=C7C=CC8=C\6C=CC=C8.Cl.O.O.O.Cl
分子式C21H21N•HCl [1.5H2O]
分子量350.9
溶解度DMF: 30 mg/mL,DMSO: 30 mg/mL,Ethanol: 30 mg/mL,Ethanol:PBS(pH 7.2) (1:1): 0.5 mg/mL
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Cyproheptadine is a first-generation antihistamine that potently antagonizes the histamine H1 receptor (pKi = 9.42). It also antagonizes serotonin and muscarinic receptors at nanomolar concentrations. Cyproheptadine also inhibits the lysine methyltransferase SET7/9 (IC50 = 1 µM), suppressing the expression of estrogen receptor α in human breast cancer MCF-7 cells.