产品名称: | 马来酸吡拉明 |
CAS: | 59-33-6 |
分子式: | C21H27N3O5 |
分子量: | 401.46 |
纯度: | >98% |
溶解性: | DMSO |
存储: | 4℃, protect from light;In solvent : -80℃, 6 months; -20℃, 1 month (protect from light) |
研究领域: | Neurological Disease;Endocrinology |
Target: | Kd: 0.8 nM (Histamine H1 receptor), 5200 nM (Histamine H2 receptor), >3000 nM (Histamine H3 receptor)[1]pKd: 9.4 (Histamine H1 receptor)[2] |
描述: | Mepyramine maleate, a first generation antihistamine, is an antagonist of histamine H1 receptor, with Kds of 0.8 nM, 5200 nM and >3000 nM for H1, H2, and H3 receptor, respectively, and a pKd of 9.4 fo |