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[Des-Arg9]-Bradykinin acetate
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
[Des-Arg9]-Bradykinin acetate图片
CAS NO:23827-91-0
包装与价格：
包装价格(元)
5mg电议
10mM (in 1mL Water)电议
25mg电议

产品介绍
[Des-Arg9]-Bradykininacetate是缓激肽B1受体(BradykininB1receptor)激动剂，对B1受体的选择性高于B2受体。
Cas No.23827-91-0
别名[Des-Arg9]-缓激肽醋酸盐
Canonical SMILESArg-Pro-Pro-Gly-Phe-Ser-Pro-Phe
分子式C46H65N11O12
分子量964.07
溶解度Water : 100 mg/mL (103.73 mM)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

[Des-Arg9]-Bradykinin acetate is a Bradykinin B1 receptor agonist that displays selectivity for B1 over B2 receptors.

[Des-Arg9]-Bradykinin acetate is a Bradykinin(B1) receptor agonist. The B2 receptor mediates the action of bradykinin (BK) and lysyl-bradykinin (Lys-BK), the first set of bioactive kinins formed in response to injury from kininogen precursors through the actions of plasma and tissue kallikreins, whereas the B1 receptor mediates the action of [Des-Arg9]-Bradykinin (des-Arg9-BK) and Lys-des-Arg Arg9-BK, the second set of bioactive kinins formed through the actions of carboxypeptidases on BK and Lys-BK, respectively[1].

[1]. Leeb-Lundberg LM, et al. International union of pharmacology. XLV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences. Pharmacol Rev. 2005 Mar;57(1):27-77.