| CAS NO: | 2361146-30-5 |
| 包装 | 价格(元) |
| 5mg | 电议 |
| 10mg | 电议 |
GSK840(GSK’840)是一种受体相互作用蛋白激酶3(RIP3orRIPK3)抑制剂，高亲和力结合RIP3激酶结构域，IC50值为0.9nM，并抑制激酶活性，IC50值为0.3nM。
| Cas No. | 2361146-30-5 |
| 别名 | GSK'840 |
| Canonical SMILES | O=C(OC(C)(C)C)CC1=CC=C(N2C3=CC=C(C(NC)=O)C=C3N=C2)C=C1 |
| 分子式 | C21H23N3O3 |
| 分子量 | 365.43 |
| 溶解度 | 110 mg/mL in DMSO |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
| 产品描述 | GSK840 (GSK’840) is a receptor-interacting protein kinase 3 (RIP3 or RIPK3) inhibitor, which binds RIP3 kinase domain with an IC50 of 0.9 nM, and inhibits kinase activity with an IC50 of 0.3 nM[1]. IC50: 0.3 nM (RIP3)[1] Reference: |
m.cnreagent.com