Acetyl-pepstatin 是一种有效的经典天冬氨酸蛋白酶 (PRs) 抑制剂,XMRV PR 和 HIV-1 PR Ki 值分别为 712 nM 和 13 nM。
Cas No. | 28575-34-0 |
别名 | 醋酸胃酶抑素,Pepstatin A acetate |
分子式 | C31H57N5O9 |
分子量 | 643.82 |
溶解度 | Soluble in DMSO |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Acetyl-pepstatin is reported to be an effective inhibitor of HIV-1 proteinase (Ki = 20 nM at pH 4.7) and of HIV-2 proteinase (Ki = 5 nM at pH 4.7). Ac-Val-Val-Sta-Ala-Sta also inhibits the P. falciparum aspartyl protease plasmepsin II, IC50 0.6 nM. |