Alprenolol((RS)-Alprenolol)

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本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

13655-52-2

包装与价格：

包装	价格(元)
10mM (in 1mL DMSO)	电议
50mg	电议
100mg	电议

产品介绍

Alprenolol ((RS)-Alprenolol) ((RS)-Alprenolol ((RS)-Alprenolol); dl-Alprenolol ((RS)-Alprenolol)) 是一种具有口服活性的非选择性 β-adrenoceptor 拮抗剂和 5 的拮抗剂-HT1A 和 5-HT1B 受体。 Alprenolol ((RS)-Alprenolol) 用作抗高血压、抗心绞痛和抗心律失常药物。

Cas No.	13655-52-2
别名	阿普洛尔; (RS)-Alprenolol; dl-Alprenolol
Canonical SMILES	OC(COC1=CC=CC=C1CC=C)CNC(C)C
分子式	C₁₅H₂₃NO₂
分子量	249.35
溶解度	DMSO : ≥ 100 mg/mL (401.04 mM);Water :< 0.1 mg/mL (insoluble)
储存条件	Store at -20°C
General tips	For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition	Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request
产品描述	Alprenolol is a non-selective beta blocker as well as 5-HT1A receptor antagonist.The reference for administration is 10 mg/kg. [1]. Schreiber R et al. Involvement of 5-HT1A receptors in the anxiolytic action of S 14671 in the pigeon conflict test. Pharmacol Biochem Behav. 1995 Jun-Jul;51(2-3):211-5. [2]. Millan MJ et al. Novel benzodioxopiperazines acting as antagonists at postsynaptic 5-HT1A receptors and as agonists at 5-HT1A autoreceptors: a comparative pharmacological characterization with proposed 5-HT1A antagonists. J Pharmacol Exp Ther, 1994 Jan, 2