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Dagrocorat(PF-00251802)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Dagrocorat(PF-00251802)图片
CAS NO:1044535-52-5
包装与价格:
包装价格(元)
250mg电议
500mg电议

产品介绍
Dagrocorat (PF-00251802) (PF-00251802) 是一种具有口服活性和选择性的糖皮质激素受体高亲和力部分激动剂。
Cas No.1044535-52-5
别名PF-00251802
Canonical SMILESO[C@@]1(C(F)(F)F)C[C@]2([H])[C@](C3=CC=C(C(NC(C=CC=N4)=C4C)=O)C=C3CC2)(CC1)CC5=CC=CC=C5
分子式C29H29F3N2O2
分子量494.55
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist.

[1]. Ripp SL,et al. In Vitro and In Vivo Investigation of Potential for Complex CYP3A Interaction for PF-00251802 (Dagrocorat), a Novel Dissociated Agonist of the Glucocorticoid Receptor. Clin Pharmacol Drug Dev. 2018 Mar;7(3):244-255.