您好,欢迎来到化工原料网! [登录] [免费注册]
化工原料网
位置:首页 > 产品库 > Epanolol(Visacor)
立即咨询
咨询类型:
     
*姓名:
*电话:
*单位:
Email:
*留言内容:
请详细说明您的需求。
*验证码:
 
Epanolol(Visacor)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Epanolol(Visacor)图片
CAS NO:86880-51-5
包装:1mg
市场价:5355元

产品介绍
Epanolol (Visacor) (Visacor; ICI141292) 是一种有效的 β-adrenoceptor 部分激动剂,对 β1- 的亲和力高于 β2-adrenoceptors。
Cas No.86880-51-5
别名依泮洛尔,Visacor; ICI141292
Canonical SMILESO=C(NCCNCC(O)COC1=CC=CC=C1C#N)CC2=CC=C(O)C=C2
分子式C20H23N3O4
分子量369.41
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Epanolol (Visacor; ICI141292) is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.

Epanolol is a novel anti-anginal agent which is a β1-adrenoceptor partial agonist exhibiting selective β1-adrenoceptor antagonist and selective β1-adrenoceptor agonist activity[1].

[1]. Hosie J, et al. Pharmacokinetics of epanolol after acute and chronic oral dosing in elderly patients with stable angina pectoris. Br J Clin Pharmacol. 1990 Mar;29(3):333-7.