CAS NO: | 86880-51-5 |
包装: | 1mg |
市场价: | 5355元 |
Cas No. | 86880-51-5 |
别名 | 依泮洛尔,Visacor; ICI141292 |
Canonical SMILES | O=C(NCCNCC(O)COC1=CC=CC=C1C#N)CC2=CC=C(O)C=C2 |
分子式 | C20H23N3O4 |
分子量 | 369.41 |
溶解度 | Soluble in DMSO |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Epanolol (Visacor; ICI141292) is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors. Epanolol is a novel anti-anginal agent which is a β1-adrenoceptor partial agonist exhibiting selective β1-adrenoceptor antagonist and selective β1-adrenoceptor agonist activity[1]. [1]. Hosie J, et al. Pharmacokinetics of epanolol after acute and chronic oral dosing in elderly patients with stable angina pectoris. Br J Clin Pharmacol. 1990 Mar;29(3):333-7. |