BPKDi 是一种有效的联吡啶PKD抑制剂,对 PKD1、PKD2 和 PKD3 的IC50分别为 1 nM、9 nM 和 1 nM。BPKDi 阻断心肌细胞中 IIa 类 HDAC 的信号依赖性磷酸化和核输出。
生物活性 | BPKDi is a potent bipyridylPKDinhibitor withIC50s of 1 nM, 9 nM and 1 nM forPKD1,PKD2andPKD3, respectively. BPKDi blocks signal-dependent phosphorylation and nuclear export of class IIa HDACs in cardiomyocytes[1]. |
IC50& Target[1] | PKD1 1 nM (IC50) | PKD2 9 nM (IC50) | PKD3 1 nM (IC50) |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |