Haspin-IN-2 (compound 4) 是一种有效的选择性的haspin抑制剂,IC50为 50 nM。Haspin-IN-1 还抑制CLK1和DYRK1A,IC50分别为 445 nM 和 917 nM。
生物活性 | Haspin-IN-2 (compound 4) is a potent and selectivehaspininhibitor with anIC50of 50 nM. Haspin-IN-1 also inbibitsCLK1andDYRK1AwithIC50s of 445 nM and 917 nM, respectively[1]. |
IC50& Target[1] | CLK1 445 nM (IC50) | DYRK1A 917 nM (IC50) | Haspin Kinase 50 nM (IC50) |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |