RMS-07 是Monopolar Spindle Kinase 1 (MPS1/TTK)的共价抑制剂,其IC50值为 13.1 nM。RMS-07靶向激酶结构域的半胱氨酸。
生物活性 | RMS-07 is a covalentMonopolar Spindle Kinase 1 (MPS1/TTK)inhibitor, with an apparentIC50of 13.1 nM. RMS-07 targets a poorly conserved cysteine in the kinase's hinge region[1]. |
IC50& Target | IC50:13.1 nM (Monopolar Spindle Kinase 1 (MPS1/TTK)). |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |