| CAS NO: | 2080311-92-6 |
| 包装 | 价格(元) |
| 100mg | 电议 |
| 250mg | 电议 |
| 500mg | 电议 |
| 生物活性 | ML233 is a non-peptide based potentapelin receptor (APJ)agonist (EC50=3.7 μM). ML233 displays >21-fold selective over the closely related angiotensin 1 (AT1) receptor (>79 μM)[1]. |
| IC50& Target | EC50: 3.7 μM (Apelin receptor)[1] |
| 体外研究 (In Vitro) | ML233 shows potentially significant binding against several other receptors, including the 5-HT1A, α2C adrenergic, and benzylpiperazine receptors and norepinephrine transporter. ML233 shows some toxicity (LC50=25.8 μM) toward human hepatocyctes[1]. |
| 分子量 | 359.44 |
| Formula | C19H21NO4S |
| CAS 号 | 2080311-92-6 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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