BI-2081 是一种GPR40 (FFAR1)部分激动剂 (EC50: 4 nM)。BI-2081 诱导葡萄糖依赖的胰岛素分泌并降低血浆葡萄糖浓度。BI-2081 可用于代谢疾病的研究,特别是 2 型糖尿病。
生物活性 | BI-2081 is aGPR40 (FFAR1)partial agonist (EC50: 4 nM). BI-2081 induces glucose dependinginsulinsecretion and reduces the plasma glucose concentration. BI-2081 can be used in the research of metabolic diseases, in particular diabetes type 2[1]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |