GRK6-IN-2 (compound 10a) is a potent inhibitor ofG protein-coupled receptor kinase 6(GRK6) with anIC₅₀of 120 nM. GRK6 is a critical kinase required for the survival of multiple myeloma (MM) cells. GRK6-IN-2 has the potential for the research of multiple myeloma^[1].

376.43

Solid

C₂₁H₂₁FN₆

2677786-27-3

Room temperature in continental US; may vary elsewhere.

Methanol : ≥ 125 mg/mL(332.07 mM)

DMSO : ≥ 100 mg/mL(265.65 mM)

*"≥" means soluble, but saturation unknown.

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储备液的保存方式和期限：-80℃, 6 months; -20℃, 1 month。-80℃ 储存时，请在 6 个月内使用，-20℃ 储存时，请在 1 个月内使用。