CAS NO: | 2410794-89-5 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | GRK5-IN-4 (Compound 16d, CCG-265328) is a potent and and selective covalentGRK5(G protein-coupled receptor kinase 5) inhibitor, with anIC50of 1.1 μM. GRK5-IN-4 shows 90-fold selectivity over GRK2. GRK5-IN-4 can be used for heart failure research[1]. |
IC50& Target | IC50: 1.1 ± 0.4 μM (GRK5), 1.8 ± 2 μM (GRK6), >100 μM (GRK2)[1] |
体外研究 (In Vitro) | GRK5-IN-4 (Compound 16d) (0-4 h) displays a marked increase in apparent potency as a function of time[1]. |
分子量 | 483.52 |
Formula | C26H25N7O3 |
CAS 号 | 2410794-89-5 |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |