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PSN 375963 hydrochloride
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
PSN 375963 hydrochloride图片
CAS NO:1781834-82-9
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品介绍
PSN 375963 hydrochloride 是一种有效的GPR119激动剂,对人和小鼠的EC50分别为 8.4 和 7.9 μM。PSN 375963 hydrochloride 显示出与内源性油酰乙醇酰胺 (OEA) 相似的效力。
生物活性

PSN 375963 hydrochloride is a potentGPR119agonist, withEC50s of 8.4 and 7.9 μM for human and mouseGPR119, respectively. PSN 375963 hydrochloride shows similar potency to the endogenous agonist oleoylethanolamide (OEA)[1][2].

体外研究
(In Vitro)

The endogenous ligand OEA signals through GPR119 in a manner similar to glucagon-like peptide-1 (GLP-1) and its receptor with respect to insulin secretion, intracellular calcium and cAMP[2].

分子量

321.84

Formula

C17H24ClN3O

CAS 号

1781834-82-9

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.