CAS NO: | 1300019-38-8 |
包装 | 价格(元) |
10 mM * 1 mL in DMSO | 电议 |
1mg | 电议 |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
200mg | 电议 |
生物活性 | I-BET762 carboxylic acid (Molibresib carboxylic acid) is an I-BET762-based warhead ligand for conjugation reactions ofPROTACtargeting on BET. I-BET762 carboxylic acid (Molibresib carboxylic acid) is aBRD4inhibitor with apIC50of 5.1[1]. | ||||||||||||||||
IC50& Target |
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体外研究 (In Vitro) | I-BET762 carboxylic acid (Molibresib carboxylic acid) (Compound 27) inhibits peripheral blood mononuclear cells (PBMC) with a pIC50of<4[1]. | ||||||||||||||||
分子量 | 396.83 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C20H17ClN4O3 | ||||||||||||||||
CAS 号 | 1300019-38-8 | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 |
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溶解性数据 | In Vitro: DMSO : 7.14 mg/mL(17.99 mM;Need ultrasonic) 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |