CTAP(trifluoroacetate salt)

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本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

包装:	1mg
市场价:	1750元

产品介绍

CTAP is a water soluble, cyclic octapeptide which acts as a receptor antagonist that is selective for the μ opioid receptor (IC50 = 3.5 nM) over the δ receptor (IC50 = 4,500 nM).

Canonical SMILES	O=C([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=C(C=C3)O)NC([C@@H](NC([C@@H](CC4=CC=CC=C4)N)=O)CSSC(C)([C@H](NC5=O)C(N[C@@H]([C@@H](C)O)C(N)=O)=O)C)=O)=O)N[C@@H](CCCNC(N)=N)C(N[C@H]5[C@@H](C)O)=O.FC(F)(C(O)=O)F
分子式	C₅₁H₆₉N₁₃O₁₁S₂•XCF₃COOH
分子量	1104.3
溶解度	Water: soluble
储存条件	Store at -20°C
General tips	For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition	Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request
产品描述	CTAP is a water soluble, cyclic octapeptide which acts as a receptor antagonist that is selective for the µ opioid receptor (IC50 = 3.5 nM) over the δ receptor (IC50 = 4,500 nM). It is a poor antagonist of the somatostatin receptor (IC50 = 14.3 μM). CTAP is at least 10-fold more potent than naltrexone as an antagonist of diverse compounds which have antinociceptive effects through the µ opioid receptor. It resists enzymatic metabolism in the blood and enters the brain and cerebrospinal fluid.