伊潘立酮代谢物 P88（P88；羟基伊潘立酮）是伊潘立酮的代谢物，伊潘立酮是一种非典型抗精神病药。
| Cas No. | 133454-55-4 |
| 别名 | 伊潘立酮代谢物; P88; Hydroxy Iloperidone |
| Canonical SMILES | OC(C)C1=CC=C(OCCCN2CCC(C3=NOC4=C3C=CC(F)=C4)CC2)C(OC)=C1 |
| 分子式 | C24H29FN2O4 |
| 分子量 | 428.5 |
| 溶解度 | Chloroform: slightly soluble,Methanol: slightly soluble |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Iloperidone metabolite P88 is an active metabolite of the atypical antipsychotic iloperidone . It binds to the serotonin (5-HT) receptor subtypes 5-HT1B, 5-HT2A, and 5-HT2C (Kis = 5.1, 0.03, and 6.9 nM, respectively), α2b- and α2c-adrenergic (Kis = 6 and 1.3 nM, respectively), and dopamine D1, D2A, and D4 receptors (Kis = 9.5, 1.6, and 3.5 nM, respectively). |
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