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PKM2 activator 3
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
PKM2 activator 3图片
CAS NO:1346113-84-5
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品介绍
PKM2 activator 3 是一种有效的PKM2激活剂,AC50为 90 nM。PKM2 activator 3 具有良好的 Caco-2 渗透性、低外排比和高微粒体稳定性。PKM2 activator 3 可用于抗癌研究。
生物活性

PKM2 activator 3 is a potentPKM2activator with anAC50value of 90 nM. PKM2 activator 3 has good Caco-2 permeability, a low efflux ratio and high microsomal stability. PKM2 activator 3 can be used for researching anticancer[1].
(AC50: the concentration which gives 50% activation of enzyme.)

IC50& Target

PKM2[1]

体内研究
(In Vivo)

PKM2 activator 3 (compound 66) has good Caco-2 permeability, a low efflux ratio (0.84) and high microsomal stability (t1/2= 277.2 min in human liver microsomes and 117.5 min in mouse liver microsomes)[1].

分子量

372.77

Formula

C15H11ClF2N2O3S

CAS 号

1346113-84-5

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.