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Dabigatran(ethyl ester)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Dabigatran(ethyl ester)图片
CAS NO:429658-95-7
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议
200mg电议
500mg电议

产品名称
达比加群乙酸乙酯
产品介绍
Dabigatran ethyl ester 是新型的口服抗凝化合物和凝血酶抑制剂。
生物活性

Dabigatran ethyl ester is an emerging oral anticoagulant which is a direct inhibitor ofthrombinactivity. IC50 value: Target:thrombinDabigatran provides a stable anticoagulation effect without any need to perform periodical laboratory controls. Of note, there is a growing amount of clinical evidence which shows its safety and efficacy. For these reasons, Dabigatran may suppose a revolution in oral anticoagulation. Dabigatran etexilate was rapidly converted to Dabigatran, with peak plasma dabigatran concentrations being attained after approximately 1.5 h; the bioavailability of Dabigatran after p.o. administration of Dabigatran etexilate was 7.2%.

分子量

499.56

性状

Solid

Formula

C27H29N7O3

CAS 号

429658-95-7

中文名称

达比加群乙酸乙酯

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式
Powder-20°C3 years
4°C2 years
In solvent-80°C6 months
-20°C1 month
溶解性数据
In Vitro: 

H2O : 1 mg/mL(2.00 mM;ultrasonic and warming and heat to 80℃)

DMSO : 1 mg/mL(2.00 mM;Need ultrasonic)

配制储备液
浓度溶剂体积质量1 mg5 mg10 mg
1 mM2.0018 mL10.0088 mL20.0176 mL
5 mM---------
10 mM---------
*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效
储备液的保存方式和期限:-80℃, 6 months; -20℃, 1 month。-80℃ 储存时,请在 6 个月内使用,-20℃ 储存时,请在 1 个月内使用。