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Obeticholic Acid-d4
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Obeticholic Acid-d4图片
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议

产品名称
奥贝胆酸 d4
产品介绍
Obeticholic Acid-d4 是 Obeticholic acid 的氘代物。Obeticholic acid (INT-747) 是一种有效的,选择性的和口服活性的FXR激动剂,EC50为 99 nM,并具有抗胆碱和抗炎作用。Obeticholic acid 还可诱导细胞自噬 (autophagy)。
生物活性

Obeticholic Acid-d4 is the deuterium labeled Obeticholic acid. Obeticholic acid (INT-747) is a potent, selective and orally activeFXRagonist with anEC50of 99 nM. Obeticholic acid has anticholeretic and anti-inflammation effect. Obeticholic acid also inducesautophagy[1][2][3].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

410.62

性状

Solid

Formula

C25H38D4O4

中文名称

奥贝胆酸 d4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式
Powder-20°C3 years
In solvent-80°C6 months
-20°C1 month