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Tauro-Obeticholic acid-d5 sodium
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Tauro-Obeticholic acid-d5 sodium图片
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品介绍
Tauro 6-Ethlchenodeoxycholic Acid-d5 (sodium salt) 是 Tauro-Obeticholic acid 氘代物。Tauro-Obeticholic acid 是牛磺酸的活性代谢物。Obeticholic Acid 是一种口服生物可利用的法尼样X受体 (FXR) 激动剂。
生物活性

Tauro 6-Ethlchenodeoxycholic Acid-d5 (sodium salt) is deuterium labeled Tauro-Obeticholic acid. Tauro-Obeticholic acid is an active metabolite of Obeticholic acid. Obeticholic acid is an orally bioavailable farnesoid-X receptor (FXR) agonist[1].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

532.79

Formula

C28H44D5NO6S

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.