CL2 Linker 是ADC分子的一种可降解 (cleavable) 的 linker。CL2-SN-38 和 CL2A-SN-38 拥有几乎等效的药物替代 (~6)、细胞结合 (Kd~1.2 nM)、细胞毒性 (IC50~2.2 nM) 以及体外血清稳定性 (t1/2~20 小时)。
生物活性 | CL2 Linker is acleavableADClinker. CL2-SN-38 and CL2A-SN-38 are equivalent in drug substitution (~6), cell binding (Kd~1.2 nM), cytotoxicity (IC50~2.2 nM), and serum stability in vitro (t1/2~20 hours)[1][2]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |