U-75302 是一种有效的白三烯 B4 抑制剂。
Cas No. | 119477-85-9 |
Canonical SMILES | OCCCC[C@H](O)CC1=NC(/C=C/[C@H](O)C/C=C\CCCCC)=CC=C1 |
分子式 | C22H35NO3 |
分子量 | 361.5 |
溶解度 | DMF: >7.1 mg/ml,DMSO: >10 mg/ml,Ethanol: >50 mg/ml,PBS 7.2: >80 µ g/ml |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | U-75302 is an LTB4 receptor antagonist with a Ki of 159 nM on guinea pig lung membranes. This activity is specific for the BLT1 receptor; U-75302 does not antagonize the binding of [3H]-LTB4 to the human BLT2 receptor. |